| Drug Name | Brand Names | Clinical Use |
| | |
| | |
| Albuterol | Ventolin, Proventil, Ecovent | Respiratory tract diseases |
| Alfuzosin | Uroxatral, Xatral | Alpha-adrenergic blocker |
| Amantadine | Symmetrel | Viral infections |
| Amiodarone | Pacerone, Cordarone | Cardiovascular diseases |
| Amitriptyline | Elavil, Tryptizol | Neuropsychiatric diseases |
| Amoxapine | Asendin | Neuropsychiatric diseases |
| Amphetamine | Adderall | Neuropsychiatric diseases |
| Arsenic trioxide | Trisenox | Cancer, leukemia |
| Atomoxetine | Strattera | Neuropsychiatric diseases |
| Azithromycin | Zithromax | Bacterial infections |
| Bepridil | Vascor | Cardiovascular diseases |
| Chloralhydrate | Noctec, Medianox | Neuropsychiatric diseases |
| Chloroquine | Arelan, Nivaquine, Chlorochin | Parasitic infections |
| Chlorpromazine | Thorazine, Chlorazin | Neuropsychiatric diseases |
| Ciprofloxacin | Ciproflox, Ciproxin | Bacterial infections |
| Cisapride | Propulsid | Gastrointestinal diseases |
| Citalopram | Celexa, Citalopram-Mepha | Neuropsychiatric diseases |
| Clarithromycin | Biaxin, Klacid | Bacterial infections |
| Clomipramine | Anafranil | Neuropsychiatric diseases |
| Clozapine | Clozaril | Neuropsychiatric diseases |
| Cocaine | Cocaine | Local anesthetic |
| Desipramine | Pertofrane | Neuropsychiatric diseases |
| Dextroamphetamine | Dexadrine | Neuropsychiatric diseases |
| Disopyramide | Norpace | Cardiovascular diseases |
| Dobutamine | Dobutrex | Cardiovascular diseases |
| Dofetilide | Tikosyn | Cardiovascular diseases |
| Dolasetron | Anzemet | Gastrointestinal diseases |
| Domperidone | Motilium | Gastrointestinal diseases |
| Dopamine | Intropine | Cardiovascular diseases |
| Doxepin | Sinquan | Neuropsychiatric diseases |
| Droperidol | Inapsine | Neuropsychiatric diseases |
| Ephedrine | Broncholate, Rynatuss | Cardiovascular diseases |
| Epinephrine | Primatene, Bronkaid | Cardiovascular diseases |
| Erythromycin | Erythrocin, Karex | Bacterial infections |
| Felbamate | Felbatrol, Taloxa | Neuropsychiatric diseases |
| Fenfluramine | Pondimin | Appetite suppressant |
| Flecainide | Tambocor | Cardiovascular diseases |
| Fluconazole | Diflucan | Fungal infections |
| Fluoxetine | Sarafem, Prozac, Fluctine | Neuropsychiatric diseases |
| Flupentixol | Fluanxol, Deanxit | Neuropsychiatric diseases |
| Foscarnet | Foscavir | Viral infections |
| Fosphenytoin | Cerebyx | Neuropsychiatric diseases |
| Galantamine | Reminyl | Neuropsychiatric diseases |
| Gatifloxacin | Tequin | Bacterial infections |
| Gemifloxacin | Factive | Bacterial infections |
| Granisetron | Kytril | Gastrointestinal diseases |
| Halofantrine | Halfan | Malaria infections |
| Haloperidol | Haldol, Sigaperidol | Neuropsychiatric diseases |
| Ibutilide | Corvert | Cardiovascular diseases |
| Imipramine | Norfranil, Tofranil | Neuropsychiatric diseases |
| Indapamide | Lozol, Fludapamid | Cardiovascular diseases |
| Isoproterenol | Isupres, Medihaler-Iso | Allergic reactions |
| Isradipine | Dynacirc, Lomir | Cardiovascular diseases |
| Itraconazole | Sporanox | Fungal infections |
| Ketoconazole | Nizoral | Fungal infections |
| Levalbuterol | Xopenex | Respiratory tract diseases |
| Levofloxacin | Levaquin, Tavanic | Bacterial infections |
| Levomethadyl | Orlaam | Neuropsychiatric diseases |
| Lithium | Eskalith, Lithobid, Priadel | Neuropsychiatric diseases |
| Mefloquin | Lariam, Mephaquin | Parasitic infections |
| Mesoridazine | Serentil | Neuropsychiatric diseases |
| Metaproterenol | Alupent, Metaprel | Respiratory tract diseases |
| Methadone | Dolophine, Methadose, Ketalgin | Neuropsychiatric diseases |
| Methylphenidate | Ritalin, Concerta | Neuropsychiatric diseases |
| Mexiletine | Mexitil | Cardiovascular diseases |
| Midodrine | Proamatine, Gutron | Cardiovascular diseases |
| Moexipril | Uniretic | High blood pressure |
| Moxifloxacin | Avelox | Bacterial infections |
| Nicardipine | Cardene | High blood pressure |
| Norepinephrine | Levophed, Scandonest | Cardiovascular diseases |
| Nortriptyline | Pamelor, Nortrilen | Neuropsychiatric diseases |
| Octreotide | Sandostatin | Carcinoid diseases |
| Ofloxacin | Floxin, Tarivid | Bacerial infections |
| Olanzapin | Zyprexa | Neuropsychiatric diseases |
| Ondansetron | Zofran | Gastrointestinal diseases |
| Paroxetine | Paxil, Deroxat, Parexat | Neuropsychiatric diseases |
| Pentamidine | Nebupent, Pentam, Pentacarinat | Pneumonia |
| Phentermine | Fastin, Adipex | Appetite suppressant |
| Phenylephrine | Neosynephrine | Asthma |
| Phenylpropanolamine | Acutrim, Dexatrim, Rhinotussal | Asthma |
| Pimozide | Orap | Neuropsychiatric diseases |
| Procainamide | Pronestyl, Procan | Cardiovascular diseases |
| Protriptyline | Vivactil | Neuropsychiatric diseases |
| Pseudoephedrine | Otrinol, Sudafed, Benical | Asthma |
| Quetiapine | Seroquel | Neuropsychiatric diseases |
| Quinidine | Quinaglute, Cardioquin | Cardiovascular diseases |
| Ranolazine | Ranexa | Chronic angina |
| Risperidone | Risperdal | Neuropsychiatric diseases |
| Ritodrine | Yutopar | Uterine relaxant |
| Roxithromycin | Rulide | Bacterial infections |
| Salmeterol | Serevent, Seretide | Respiratory tract diseases |
| Sertindol | Serdolect | Neuropsychiatric diseases |
| Sertraline | Zoloft, Gladem | Neuropsychiatric diseases |
| Sibutramine | Meridia, Ionamine | Appetite suppressant |
| Solifenacin | Vesicare | Neuropsychiatric diseases |
| Sotalol | Betapace, Sotalex | Cardiovascular diseases |
| Sparfloxacin | Zagam | Bacterial infections |
| Tacrolimus | Prograf, Protopic | Immune suppression |
| Tamoxifen | Nolvadex | Breast cancer |
| Telithromycin | Ketek | Bacterial infections |
| Terbutaline | Brethine, Bricanyl | Respiratory tract diseases |
| Thioridazine | Mellaril, Melleretten | Neuropsychiatric diseases |
| Tizanidine | Zanaflex | Muscle relaxant |
| Tolterodine | Detrol | Bladder antispasmodic |
| Trimethoprim-Sulfa | Sulfa, Bactrim, Cotrim | Bacterial infections |
| Trimipramine | Surmontil, Trimin | Neuropsychiatric diseases |
| Vardenafil | Levitra | Phosphodiesterase inhibitor |
| Venlafaxine | Effexor | Neuropsychiatric diseases |
| Voriconazole | Vfend | Fungal infections |
| Ziprasidone | Geodon | Neuropsychiatric diseases |